Supporting Information Discovery of N-phenyl-4-(thiazol-5-yl)pyrimidin- 2-amine Aurora Kinase Inhibitors
نویسندگان
چکیده
Supporting Figure 1. Kinase inhibitory activity of compound 18 . S2 Supporting Figure 2. Activity of compound 18 in tumor models S3 Synthesis and Characterization of Compounds 7h, 11–17, and 19–24 S4 Biopharmaceutical Profiling S7 Rat Pharmacokinetics S7 Cell Viability Assay S7 Murine P388/D1 Leukemia Model S7 NCI-H460 Xenograft S7 X-Ray Crystallography S8 Molecular Modeling S8 Supplementary References S8
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